SCHEMBL1096776

SCHEMBL1096776

C[C@H](c1cccc2ccccc12)N(CC1CCN(C(N)=S)CC1c1cccc(F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.39
KCNH2 Q12809 2/20 0.35
GPR119 Q8TDV5 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1105750 0.90 CCR5 (0.40) CCR5KCNH2GPR119ESR1ESR2
SCHEMBL3576540 0.89 CCR5 (0.39) CCR5KCNH2
SCHEMBL1095663 0.88 CCR5 (0.40) CCR5KCNH2
SCHEMBL1097652 0.86 CCR5 (0.38) CCR5KCNH2GPR119
SCHEMBL1096057 0.85 CCR5 (0.38) CCR5GPR119
SCHEMBL1096778 0.84 CCR5 (0.39) CCR5KCNH2
SCHEMBL1096420 0.84 CCR5 (0.36) CCR5GPR119ESR1ESR2
SCHEMBL1097046 0.83 CCR5 (0.37) CCR5KCNH2
SCHEMBL1096488 0.83 CCR5 (0.39) CCR5ESR1ESR2
SCHEMBL1096227 0.83 CCR5 (0.36) CCR5GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153658-B2 Piperidine derivative or salt thereof ASTELLAS PHARMA, INC. (JP) 2012-04-10 US disclosed