SCHEMBL10976299

SCHEMBL10976299

CC(=O)c1ccc(Cl)cc1-c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.52
MKNK1 Q9BUB5 2/20 0.50
MKNK2 Q9HBH9 2/20 0.50
KCNMA1 Q12791 1/20 0.50
CNR1 P21554 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
KLK7 P49862 1/20 0.47
CLK1 P49759 1/20 0.47
DYRK1A Q13627 1/20 0.47
CYP2C9 P11712 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2A6 P11509 2/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3515912 0.84 CFTR (0.53) CYP11B2MKNK1MKNK2KCNMA1CNR1
SCHEMBL18057577 0.82 PTGDR2 (0.50) MEN1KMT2AMAPTCYP2C19
Acetic Acid SCHEMBL27950053 0.81 MEN1 (0.48) CYP11B2MKNK1MKNK2CNR1MEN1
SCHEMBL9206961 0.79 CYP2A6 (0.53) MKNK1MKNK2KMT2AMAPTCYP2C9
SCHEMBL8940388 0.79 P2RX1 (0.46) CNR1MEN1KMT2AMAPT
SCHEMBL14439661 0.78 ALDH1A1 (0.48) MEN1KMT2AMAPTMAPK1
SCHEMBL16574106 0.78 CYP2A6 (0.51) CYP11B2CNR1MEN1KMT2ACYP2C9
SCHEMBL7582709 0.77 CYP2A6 (0.53) CYP11B2MKNK1MKNK2CNR1MAPT
SCHEMBL28115752 0.76 CYP2A6 (0.51) CYP11B2CNR1MEN1KMT2AMAPT
SCHEMBL16982975 0.74 CYP2A6 (0.51) CYP11B2CNR1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0049854-B1 PYRIDINE AND PYRAZINE DERIVATIVES, PREPARATION OF THESE COMPOUNDS, FUNGICIDAL AGENTS CONTAINING THESE COMPOUNDS AS ACTIVE INGREDIENTS, AND THE USE OF SUCH COMPOUNDS OR AGENTS AS FUNGICIDES IN AGRICULTURE AND IN HORTICULTURE F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-01-16 EP disclosed