SCHEMBL10977484

SCHEMBL10977484

CN(C(=O)c1cccnc1Oc1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 15/20 0.55
KDM4E B2RXH2 1/20 0.54
MEN1 O00255 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C19 P33261 1/20 0.54
KMT2A Q03164 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
GPBAR1 Q8TDU6 1/20 0.53
RXFP1 Q9HBX9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10972225 0.92 KDM4E (0.60) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL29991644 0.83 MEN1 (0.63) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL2333429 0.83 MEN1 (0.63) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL30166677 0.83 MEN1 (0.63) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL30792433 0.81 KMT2A (0.62) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL9122123 0.80 TDP1 (0.66) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL8177633 0.79 KDM4E (0.62) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL10969027 0.79 KDM4E (0.62) P2RY1KDM4EMEN1CYP1A2CYP2C19
SCHEMBL4302001 0.79 KMT2A (0.49) KDM4EMEN1KMT2AGPBAR1RXFP1
O-Xylene SCHEMBL28789870 0.78 KDM4E (0.56) P2RY1KDM4EMEN1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0053011-A1 New herbicidal nicotinamide derivatives MAY & BAKER LIMITED (GB) 1982-06-02 EP claimed
EP-0053011-B1 NEW HERBICIDAL NICOTINAMIDE DERIVATIVES MAY & BAKER LIMITED (GB) 1985-04-03 EP disclosed
EP-0053011-A1 New herbicidal nicotinamide derivatives MAY & BAKER LIMITED (GB) 1982-06-02 EP disclosed