SCHEMBL10977488

SCHEMBL10977488

COc1ccc(-c2cnc(N(Cc3ccccc3)c3ccccc3)nc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
CYP19A1 P11511 1/20 0.43
NOS1 P29475 1/20 0.42
MAPK1 P28482 1/20 0.42
LTA4H P09960 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
G6PC1 P35575 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
EGFR P00533 1/20 0.41
CSF1R P07333 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
OXTR P30559 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10972930 0.86 TP53 (0.47) CYP19A1EGFRCSF1RNPC1RAB9A
SCHEMBL10972922 0.84 MCHR1 (0.43) TRPM8EGFRNPC1RAB9AOXTR
SCHEMBL10973834 0.80 KDR (0.45) LMNANPC1RAB9AL3MBTL1
SCHEMBL27827514 0.79 LTA4H (0.55) TSHRMAPK1LTA4HLMNAG6PC1
SCHEMBL10977769 0.79 MERTK (0.46) EGFRCSF1RNPC1RAB9A
SCHEMBL8908075 0.77 LTA4H (0.57) TSHRLTA4HG6PC1TRPM8
SCHEMBL899366 0.77 HSD17B2 (0.46) TSHRNOS1MAPK1LMNASMN1; SMN2
SCHEMBL10971330 0.75 KDR (0.41) LMNATRPM8EGFRNPC1RAB9A
SCHEMBL11876127 0.73 BCHE (0.53) TSHRLTA4HSMN1; SMN2NPC1RAB9A
SCHEMBL6486634 0.73 CYP2C19 (0.58) TSHRCYP19A1MAPK1LTA4HLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-85103378-A Process for preparing a group of novel compounds, formulations containing these compounds and their use in therapy 1986-07-09 CN claimed
EP-0164204-A1 Novel pharmaceutically useful pyrimidines FISONS plc (GB) 1985-12-11 EP claimed