SCHEMBL10983294

SCHEMBL10983294

CC(=Cc1ccc(Sc2ccncc2)cc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.53
TBXAS1 P24557 9/20 0.48
DDAH1 O94760 1/20 0.45
NOS1 P29475 1/20 0.45
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE7A Q13946 1/20 0.39
AKR1C2 P52895 2/20 0.39
AKR1C1 Q04828 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NEK2 P51955 1/20 0.37
PLK1 P53350 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10983292 1.00 AKR1C3 (0.53) AKR1C3TBXAS1DDAH1NOS1HPGD
Hydrochloric Acid SCHEMBL10989976 0.98 AKR1C3 (0.51) AKR1C3TBXAS1DDAH1NOS1HPGD
Hydrochloric Acid SCHEMBL10989978 0.98 AKR1C3 (0.51) AKR1C3TBXAS1DDAH1NOS1HPGD
SCHEMBL7268646 0.84 AKR1C3 (0.67) AKR1C3TBXAS1CYP1A2CYP3A4CYP2D6
SCHEMBL7963228 0.84 AKR1C3 (0.67) AKR1C3TBXAS1CYP1A2CYP3A4CYP2D6
SCHEMBL27224536 0.84 AKR1C3 (0.67) AKR1C3TBXAS1CYP1A2CYP3A4CYP2D6
SCHEMBL8374501 0.79 PDE7A (0.39) AKR1C3TBXAS1PDE7A
SCHEMBL8441479 0.79 PDE7A (0.39) AKR1C3TBXAS1PDE7A
SCHEMBL2462983 0.78 AKR1C3 (0.82) AKR1C3TBXAS1L3MBTL1ALDH1A1
SCHEMBL2462984 0.78 AKR1C3 (0.82) AKR1C3TBXAS1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4496735-A THROMBOXANE A2 INHIBITOR MARUKO SEIYAKU CO., LTD. (JP) 1985-01-29 US claimed
US-4496735-A THROMBOXANE A2 INHIBITOR MARUKO SEIYAKU CO., LTD. (JP) 1985-01-29 US disclosed