SCHEMBL10990752

SCHEMBL10990752

Cc1cccc(C)c1NC(=O)CN1CCN(CC(O)C2COc3c(ccc(Cl)c3C)O2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
ADRB1 P08588 2/20 0.45
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1A P35348 2/20 0.45
DRD3 P35462 2/20 0.45
HTR2B P41595 2/20 0.45
KCNH2 Q12809 2/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
ADRB2 P07550 1/20 0.45
SCN5A Q14524 1/20 0.45
LMNA P02545 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
DRD4 P21917 3/20 0.41
ALDH1A1 P00352 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10995598 0.90 CYP3A4 (0.43) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL7440560 0.88 ALDH1A1 (0.45) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10997730 0.86 CYP3A4 (0.47) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10997843 0.85 CYP3A4 (0.45) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10990432 0.85 CYP3A4 (0.45) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10990695 0.85 CYP3A4 (0.52) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL10987535 0.84 LMNA (0.52) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10992935 0.84 CYP3A4 (0.48) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10996846 0.83 CYP3A4 (0.47) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL10994557 0.83 CYP3A4 (0.47) CYP3A4CYP2D6ADRB1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed