SCHEMBL10995571

SCHEMBL10995571

CCc1nc(N)nc(N)c1-c1ccc(N)c(Cl)c1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 4/20 0.68
HEXB P07686 4/20 0.68
DHFR P00374 3/20 0.68
MEN1 O00255 1/20 0.68
SLC22A1 O15245 1/20 0.68
ALDH1A1 P00352 1/20 0.68
LMNA P02545 1/20 0.68
TP53 P04637 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
HTR1A P08908 1/20 0.68
ADRA2A P08913 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C9 P11712 1/20 0.68
HTR2A P28223 1/20 0.68
ADRA1A P35348 1/20 0.68
HTR2B P41595 1/20 0.68
SLC6A3 Q01959 1/20 0.68
KMT2A Q03164 1/20 0.68
PDE4D Q08499 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etoprine SCHEMBL3919 0.90 DHFR (0.70) HEXAHEXBDHFRMEN1SLC22A1
SCHEMBL8903514 0.88 DHFR (0.68) HEXAHEXBDHFRMEN1SLC22A1
SCHEMBL6361050 0.84 HEXA (0.68) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL25129 0.81 HEXA (1.00) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL29381161 0.81 HEXA (1.00) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL15516970 0.81 HEXA (1.00) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL11709944 0.80 HEXA (0.97) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL28347069 0.80 HEXA (0.97) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL28861797 0.80 HEXA (0.97) HEXAHEXBDHFRMEN1SLC22A1
Pyrimethamine SCHEMBL8086889 0.80 HEXA (0.97) HEXAHEXBDHFRMEN1SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147443-A1 PYRIMIDINE DERIVATIVES Aston Molecules Limited (GB) 1985-07-10 EP disclosed
WO-1984004746-A1 PYRIMIDINE DERIVATIVES UNIV BIRMINGHAM (GB) 1984-12-06 WO disclosed