SCHEMBL10998627

SCHEMBL10998627

Nc1cnc(N2CCOCC2)nc1O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.52
PIK3CD O00329 2/20 0.52
PIK3CB P42338 2/20 0.52
KDM4E B2RXH2 2/20 0.51
PIK3R1 P27986 6/20 0.49
MTOR P42345 6/20 0.49
POLB P06746 1/20 0.49
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPK1 P28482 1/20 0.48
PTPN11 Q06124 1/20 0.47
TSHR P16473 1/20 0.47
GAA P10253 1/20 0.44
MAP3K12 Q12852 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10999945 0.84 ALDH1A1 (0.45) PIK3CAPIK3CDPIK3CBKDM4EPOLB
SCHEMBL10998112 0.83 SMN1; SMN2 (0.46) KDM4EPOLBALDH1A1MAPK1PTPN11
SCHEMBL27586071 0.83 KDM4E (0.54) PIK3CAPIK3CDPIK3CBKDM4EPIK3R1
SCHEMBL11002348 0.80 PTPN11 (0.47) PIK3CAPIK3CDPIK3CBKDM4EPOLB
SCHEMBL11002487 0.80 ALDH1A1 (0.44) KDM4EKMT2AALDH1A1TSHR
SCHEMBL11000227 0.80 MAPT (0.55) POLBKMT2AALDH1A1MAPK1PTPN11
SCHEMBL10995352 0.78 CDK1 (0.40) PIK3CAPIK3CDPIK3CBKDM4EMTOR
SCHEMBL10996681 0.78 PIK3CD (0.32) PIK3CAPIK3CDPIK3CBPOLBALDH1A1
SCHEMBL10328269 0.76 PIK3CA (0.64) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL10996942 0.76 PTPN11 (0.36) KDM4EPOLBALDH1A1MAPK1PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE31926-E Penicillins and salts thereof BOEHRINGER INGELHEIM GMBH (DE) 1985-06-25 US disclosed
EP-0003814-B1 PENICILLINS, THEIR SALTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1981-12-16 EP disclosed
US-4241056-A ANTIBIOTICS BOEHRINGER INGELHEIM GMBH (DE) 1980-12-23 US disclosed
EP-0003814-A2 Penicillins, their salts, process for their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1979-09-05 EP disclosed