SCHEMBL10998796

SCHEMBL10998796

N#Cc1cc(-c2ccnc(O)n2)c[nH]c1=O

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.57
PIK3CA P42336 1/20 0.57
PIK3CB P42338 1/20 0.57
MCL1 Q07820 8/20 0.52
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
AURKA O14965 2/20 0.43
TTK P33981 2/20 0.43
AURKB Q96GD4 2/20 0.43
INCENP Q9NQS7 2/20 0.43
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
KMO O15229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10998912 0.88 PIK3CD (0.56) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11002430 0.85 PIK3CD (0.56) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11035255 0.84 PIK3CD (0.52) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10995889 0.82 AURKA (0.67) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11000905 0.82 PIK3CD (0.52) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10999253 0.80 AURKB (0.65) KDM4EALDH1A1HPGDAURKATTK
SCHEMBL10842808 0.79 PIK3CD (0.67) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10707443 0.77 MCL1 (0.63) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11003994 0.77 AURKA (0.45) AURKATTKAURKBINCENP
SCHEMBL11000261 0.76 PIK3CD (0.55) PIK3CDPIK3CAPIK3CBMCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4514400-A Cardiotonic 5-heteroaryl-pyridone WILLIAM H. RORER, INC. (US) 1985-04-30 US disclosed