SCHEMBL11002430

SCHEMBL11002430

Cc1nccc(-c2c[nH]c(=O)c(C#N)c2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.56
PIK3CA P42336 1/20 0.56
PIK3CB P42338 1/20 0.56
MCL1 Q07820 9/20 0.51
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
AURKA O14965 2/20 0.45
TTK P33981 2/20 0.45
AURKB Q96GD4 2/20 0.45
INCENP Q9NQS7 2/20 0.45
AAK1 Q2M2I8 1/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 2/20 0.40
PDE5A O76074 1/20 0.40
TSHR P16473 1/20 0.40
PTGS1 P23219 1/20 0.40
PDE4A P27815 1/20 0.40
CYP2C19 P33261 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10998796 0.85 PIK3CD (0.57) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10998912 0.84 PIK3CD (0.56) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11000905 0.83 PIK3CD (0.52) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10995889 0.83 AURKA (0.67) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10995911 0.82 PIK3CD (0.52) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL11035255 0.81 PIK3CD (0.52) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10999252 0.79 AURKB (0.69) KDM4EALDH1A1HPGDAURKATTK
SCHEMBL10842808 0.78 PIK3CD (0.67) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10707443 0.76 MCL1 (0.63) PIK3CDPIK3CAPIK3CBMCL1KDM4E
SCHEMBL10998400 0.76 PIK3CD (0.49) PIK3CDPIK3CAPIK3CBMCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4514400-A Cardiotonic 5-heteroaryl-pyridone WILLIAM H. RORER, INC. (US) 1985-04-30 US disclosed