SCHEMBL10999972

SCHEMBL10999972

O=C1C(=O)N(Cc2ccc(Cl)c(Cl)c2)c2c(F)cccc21

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 5/20 0.71
ALDH1A1 P00352 7/20 0.65
APAF1 O14727 3/20 0.65
BCHE P06276 2/20 0.65
CES1 P23141 2/20 0.65
TP53 P04637 1/20 0.65
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
MAPT P10636 1/20 0.65
ALOX15 P16050 1/20 0.65
TSHR P16473 1/20 0.65
ALOX12 P18054 1/20 0.65
ACHE P22303 1/20 0.65
HSD17B10 Q99714 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
ALDH3A1 P30838 6/20 0.61
CHRM3 P20309 1/20 0.57
CA12 O43570 2/20 0.51
CA9 Q16790 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12930211 0.84 CHRM5 (0.76) CHRM5ALDH1A1CES1ACHEALDH3A1
SCHEMBL11008095 0.83 CHRM5 (0.64) CHRM5ALDH1A1APAF1BCHECES1
SCHEMBL5426477 0.79 ALDH1A1 (1.00) CHRM5ALDH1A1APAF1BCHECES1
SCHEMBL29487533 0.79 ALDH1A1 (1.00) CHRM5ALDH1A1APAF1BCHECES1
SCHEMBL30081910 0.79 ALDH1A1 (1.00) CHRM5ALDH1A1APAF1BCHECES1
SCHEMBL12930254 0.76 CHRM5 (0.61) CHRM5ALDH1A1TP53MAPTALDH3A1
SCHEMBL18668985 0.76 ALDH1A1 (0.70) ALDH1A1APAF1BCHECES1TP53
SCHEMBL22589199 0.76 ALDH1A1 (1.00) CHRM5ALDH1A1ALDH3A1
SCHEMBL10979016 0.76 ALDH1A1 (0.69) CHRM5ALDH1A1APAF1BCHECES1
SCHEMBL28026196 0.76 CHRM5 (0.72) CHRM5ALDH1A1APAF1BCHECES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4544662-A ALDOSE REDUCTASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES (GB) 1985-10-01 US disclosed
EP-0094184-A1 Indoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-16 EP disclosed