SCHEMBL11001094

SCHEMBL11001094

COC(=O)[C@H](CC(=O)OC(C)(C)C)NC1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.37
CACNA1B Q00975 5/20 0.35
CYP2C9 P11712 1/20 0.35
NPR3 P17342 1/20 0.35
CYP2C19 P33261 1/20 0.35
CA12 O43570 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
POLB P06746 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
EPHX1 P07099 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38032 0.94 EPHX1 (0.40) CYP2D6CACNA1BITGB3ITGA2BHDAC1
SCHEMBL38034 0.94 EPHX1 (0.40) CYP2D6CACNA1BITGB3ITGA2BHDAC1
SCHEMBL38058 0.80 EPHX1 (0.40) CYP2D6CACNA1BHDAC3HDAC1HDAC2
SCHEMBL38057 0.80 EPHX1 (0.40) CYP2D6CACNA1BHDAC3HDAC1HDAC2
SCHEMBL10825239 0.79 EPHX1 (0.43) CYP2D6CACNA1BHDAC3HDAC1HDAC2
SCHEMBL19744864 0.79 EPHX1 (0.43) CYP2D6CACNA1BHDAC3HDAC1HDAC2
SCHEMBL7432656 0.79 EPHX2 (0.42) CYP2C9NPR3CYP2C19POLBSMN1; SMN2
SCHEMBL7432662 0.79 EPHX2 (0.42) CYP2C9NPR3CYP2C19POLBSMN1; SMN2
SCHEMBL25076244 0.78 KMT2A (0.39) CYP2C9NPR3CYP2C19CA12POLB
SCHEMBL15075041 0.76 CYP2D6 (0.54) CYP2D6CACNA1BCYP2C9CYP2C19CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0135429-A1 The synthesis of cyclopropane amino acids and peptides THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1985-03-27 EP disclosed