SCHEMBL11003142

SCHEMBL11003142

CSc1ccc(-c2cc(C#N)c(=O)[nH]c2C)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.69
HPGD P15428 3/20 0.69
ALDH1A1 P00352 2/20 0.69
GALR3 O60755 1/20 0.69
GAA P10253 1/20 0.69
PDE3A Q14432 8/20 0.66
PDE3B Q13370 7/20 0.66
PDE4A P27815 3/20 0.66
BLM P54132 2/20 0.66
PDE4B Q07343 2/20 0.66
PDE4C Q08493 2/20 0.66
PDE4D Q08499 2/20 0.66
PDE5A O76074 1/20 0.66
LMNA P02545 1/20 0.66
TSHR P16473 1/20 0.66
PTGS1 P23219 1/20 0.66
CYP2C19 P33261 1/20 0.66
PDE2A O00408 1/20 0.56
PDE1A P54750 1/20 0.56
PDE1B Q01064 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11006744 0.85 HPGD (0.64) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL8210361 0.84 KDM4E (0.75) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL5470727 0.82 HPGD (0.73) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL9587750 0.82 KDM4E (0.73) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL10891425 0.82 KDM4E (0.73) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL7407595 0.82 KDM4E (0.73) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL11002221 0.82 PDE3A (0.68) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL5460125 0.82 KDM4E (1.00) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL11020496 0.81 MEN1 (0.77) KDM4EHPGDALDH1A1GALR3GAA
SCHEMBL8092522 0.80 GCGR (0.53) KDM4EHPGDALDH1A1GALR3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4517192-A 6-Alkyl-5-[4-(alkylsulfinyl or alkylsulfonyl)phenyl]-2(1H)-pyridinones and their use as cardiatonics STERLING DRUG INC. (US) 1985-05-14 US disclosed