SCHEMBL11005174

SCHEMBL11005174

COc1c(NCC#N)cccc1-c1nc2cncnc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.32
CYP1A2 P05177 6/20 0.32
CYP3A4 P08684 6/20 0.32
CYP2D6 P10635 5/20 0.32
CYP2C19 P33261 5/20 0.32
FGFR1 P11362 1/20 0.31
FGFR2 P21802 1/20 0.31
TYK2 P29597 1/20 0.31
FGFR3 P22607 1/20 0.31
PIK3CD O00329 1/20 0.31
EGFR P00533 1/20 0.31
TSHR P16473 4/20 0.31
CLK4 Q9HAZ1 4/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GUSB P08236 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11011418 0.89 PDE5A (0.32) PDE5ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11007757 0.84 MAPT (0.34) PDE5ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11005181 0.84 METAP2 (0.40) PDE5AFGFR1FGFR2TYK2
SCHEMBL11011531 0.83 FGFR1 (0.38) PDE5ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11010987 0.81 KDM4E (0.39) PDE5AFGFR1FGFR2FGFR3TSHR
SCHEMBL11009966 0.77 PIK3CD (0.35) PDE5ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11011131 0.77 MAOB (0.39) PDE5ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11010174 0.77 CYP17A1 (0.39) PDE5APIK3CD
SCHEMBL11007618 0.75 PDE5A (0.31) PDE5AFGFR1FGFR2ALDH1A1
SCHEMBL11007368 0.74 FGFR1 (0.38) PDE5ACYP1A2CYP3A4FGFR1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed