SCHEMBL11005642

SCHEMBL11005642

COc1ccc2c(c1)C(O)CS2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
RYR2 Q92736 7/20 0.40
KCNH2 Q12809 1/20 0.40
LMNA P02545 1/20 0.39
KDM4E B2RXH2 2/20 0.37
HTT P42858 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.36
SNCA P37840 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.36
APP P05067 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11463305 0.73 HSD17B3 (0.48) MAOAMAOBRYR2KCNH2KDM4E
SCHEMBL25659971 0.71 RYR2 (0.45) MAOAMAOBRYR2KCNH2LMNA
SCHEMBL11003635 0.71 CYP3A4 (0.36) MAOAALDH1A1KMT2A
SCHEMBL11002734 0.69 RYR2 (0.46) RYR2KCNH2KDM4EHTTPTGDR2
SCHEMBL11342238 0.68 RAD52 (0.40) HTTHTR2CHTR2BHTR2ASNCA
SCHEMBL18287927 0.67 ALDH1A1 (0.44) MAOAKDM4EHTR2ASNCAALDH1A1
SCHEMBL9565814 0.67 ALDH1A1 (0.40) ALDH1A1NPC1MEN1MAPTKMT2A
SCHEMBL9730758 0.67 RYR2 (0.44) RYR2KCNH2MTNR1A
SCHEMBL9085563 0.67 DRD2 (0.54) RYR2KCNH2
SCHEMBL1686617 0.67 KDM1A (0.42) MAOAMAOBKDM4EHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4537976-A Benzo[b]thiophenes HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1985-08-27 US disclosed
US-4528399-A Benzo[b]thiophenes intermediates HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1985-07-09 US disclosed
US-4436748-A HYPOTENSIVES, DIURETICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1984-03-13 US disclosed
EP-0050326-A2 Benzo(b)thiophenes HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1982-04-28 EP disclosed