SCHEMBL11006451

SCHEMBL11006451

O=C(Nc1cc(Cl)c(Cl)c(Cl)c1)Nc1cc(Cl)c(Cl)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.61
EPHX2 P34913 2/20 0.61
S1PR2 O95136 1/20 0.58
P2RY1 P47900 1/20 0.57
MEN1 O00255 10/20 0.53
KMT2A Q03164 10/20 0.53
LMNA P02545 7/20 0.53
NPC1 O15118 6/20 0.53
HTT P42858 5/20 0.53
ADORA3 P0DMS8 1/20 0.53
CHRM1 P11229 1/20 0.53
SLC6A2 P23975 1/20 0.53
PDE4A P27815 1/20 0.53
ADRA1A P35348 1/20 0.53
OPRM1 P35372 1/20 0.53
PDE3A Q14432 1/20 0.53
NLRP3 Q96P20 1/20 0.53
MAPT P10636 7/20 0.50
RAB9A P51151 5/20 0.50
SLC2A1 P11166 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12499941 0.91 P2RY1 (0.70) EPHX1EPHX2S1PR2P2RY1MEN1
SCHEMBL11007336 0.88 KMT2A (0.70) EPHX1EPHX2MEN1KMT2ALMNA
SCHEMBL6567241 0.83 EPHX1 (0.59) EPHX1EPHX2S1PR2P2RY1MEN1
SCHEMBL2097416 0.83 EPHX1 (0.43) EPHX1EPHX2S1PR2P2RY1MEN1
SCHEMBL2097418 0.83 THRA (0.44) EPHX1EPHX2S1PR2P2RY1MEN1
SCHEMBL20535682 0.81 LMNA (0.56) MEN1KMT2ALMNAHTTMAPT
SCHEMBL11005058 0.78 KDR (0.85) EPHX1EPHX2CA2CA9KDR
SCHEMBL15786287 0.77 MEN1 (0.76) EPHX1EPHX2S1PR2P2RY1MEN1
SCHEMBL11001550 0.77 MEN1 (0.74) EPHX1EPHX2P2RY1MEN1KMT2A
SCHEMBL9349095 0.76 KMT2A (0.48) EPHX1EPHX2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015110-A2 Anticoccidial composition, carbanilides and method of preparing them ELI LILLY AND COMPANY (US) 1980-09-03 EP claimed
US-11583509-B2 Compound for treating cancer and diabetes CITY OF HOPE (US) 2023-02-21 US disclosed
US-20220023240-A1 COMPOUND FOR TREATING CANCER AND DIABETES CITY OF HOPE 2022-01-27 US disclosed
US-9808434-B2 Compound for treating cancer and diabetes CITY OF HOPE (US) 2017-11-07 US disclosed
US-20160354327-A1 COMPOUND FOR TREATING CANCER AND DIABETES CITY OF HOPE 2016-12-08 US disclosed
US-20140162996-A1 NOVEL MODULATORS OF DEVELOPMENT OF ADIPOCYTE AND CANCER CELLS CITY OF HOPE (US) 2014-06-12 US disclosed
EP-0015110-B1 ANTICOCCIDIAL COMPOSITION, CARBANILIDES AND METHOD OF PREPARING THEM ELI LILLY AND COMPANY (US) 1985-08-21 EP disclosed
US-4526997-A Amino, nitro, fluoro substituted carbanilides DOHERTY GEORGE O P O 1985-07-02 US disclosed
US-4468380-A Anticoccidial combinations comprising polyether antibiotics and carbanilides ELI LILLY AND COMPANY (US) 1984-08-28 US disclosed
EP-0015110-A2 Anticoccidial composition, carbanilides and method of preparing them ELI LILLY AND COMPANY (US) 1980-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220023240-A1 COMPOUND FOR TREATING CANCER AND DIABETES TP53, VHL, SLC2A4 EPHX1 3055/4885EPHX2 3211/4885S1PR2 4184/4885
US-11583509-B2 Compound for treating cancer and diabetes TP53, VHL, SLC2A4 EPHX1 3055/4885EPHX2 3211/4885S1PR2 4184/4885
US-20160354327-A1 COMPOUND FOR TREATING CANCER AND DIABETES TP53, VHL, SLC2A4 EPHX1 3055/4885EPHX2 3211/4885S1PR2 4184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.