SCHEMBL11007015

SCHEMBL11007015

COc1cc2c3c(c1OC)CN(C)CC3c1ccccc1CC2

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.50
SLC6A4 P31645 11/20 0.50
SLC6A3 Q01959 8/20 0.50
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
DRD1 P21728 4/20 0.44
DRD2 P14416 2/20 0.44
PNPLA2 Q96AD5 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR7 P34969 1/20 0.44
DRD5 P21918 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11014045 0.87 DRD2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL11005867 0.86 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL11015653 0.86 DRD1 (0.39) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL11008872 0.86 DRD1 (0.39) SLC6A2SLC6A4CYP3A4CYP2D6DRD1
SCHEMBL11014467 0.83 BCHE (0.44)
SCHEMBL11010302 0.82 DRD1 (0.48) CYP2D6DRD1DRD2PNPLA2HTR2A
SCHEMBL11011835 0.81 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL11009453 0.78 HTR2A (0.43) CYP3A4CYP2D6DRD1DRD2PNPLA2
Hydrochloric Acid SCHEMBL11006734 0.77 HTR2A (0.42) CYP3A4CYP2D6DRD1DRD2PNPLA2
Bromide SCHEMBL11010072 0.75 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3DRD1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4522946-A FREE OF EXTRA-PYRAMIDAL SIDE EFFECTS AYERST, MCKENNA & HARRISON, INC. (CA) 1985-06-11 US disclosed