SCHEMBL11007271

SCHEMBL11007271

Cc1ccc(Br)c2c1CN(NC1=NCCN1)C2

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.51
HTR1D P28221 3/20 0.43
HTR1B P28222 2/20 0.43
ADRA2C P18825 5/20 0.42
ADRA2A P08913 5/20 0.42
CFB P00751 3/20 0.42
ADRA1A P35348 2/20 0.42
KCNH2 Q12809 1/20 0.42
ADRA2B P18089 4/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1B P35368 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11007474 0.92 NISCH (0.58) NISCHHTR1DHTR1BADRA2CADRA2A
SCHEMBL10767501 0.92 NISCH (0.58) NISCHHTR1DHTR1BADRA2CADRA2A
SCHEMBL10765153 0.84 NISCH (0.51) NISCHHTR1DHTR1BADRA2CADRA2A
SCHEMBL11001474 0.78 NISCH (0.72) NISCHHTR1DADRA2CADRA2AADRA1A
SCHEMBL11428144 0.74 NISCH (0.55) NISCHHTR1DHTR1BADRA2CADRA2A
SCHEMBL10764582 0.74 NISCH (0.74) NISCHHTR1DHTR1BADRA2CADRA2A
SCHEMBL11003828 0.73 NISCH (0.54) NISCHHTR1DADRA2CADRA2AADRA1A
SCHEMBL10765612 0.73 NISCH (0.54) NISCHADRA2CADRA2AADRA1AADRA2B
SCHEMBL11006239 0.71 NISCH (0.52) NISCHHTR1DADRA2CADRA2AADRA2B
SCHEMBL6054462 0.70 NISCH (0.69) NISCHADRA2CADRA2AADRA1AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4526897-A Hypertensive agents BEIERSDORF AKTIENGESELLSCHAFT (DE) 1985-07-02 US disclosed
EP-0072954-A2 Isoindolin-2-yl-amino-imidazolines and isoindolin-2-yl guanidines, process for their preparation and their use as medicines Beiersdorf Aktiengesellschaft (DE) 1983-03-02 EP disclosed