SCHEMBL11006239

SCHEMBL11006239

CCCc1ccc(CCC)c2c1CN(NC1=NCCN1)C2

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 3/20 0.52
ADRA2B P18089 12/20 0.43
ADRA2C P18825 12/20 0.43
ADRA2A P08913 12/20 0.43
HTR1A P08908 2/20 0.39
HTR1D P28221 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10767501 0.78 NISCH (0.58) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL11007474 0.75 NISCH (0.58) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL10764582 0.75 NISCH (0.74) NISCHADRA2BADRA2CADRA2AHTR1A
SCHEMBL11003828 0.74 NISCH (0.54) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL10765612 0.74 NISCH (0.54) NISCHADRA2BADRA2CADRA2A
SCHEMBL11001474 0.71 NISCH (0.72) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL11007271 0.71 NISCH (0.51) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL6054462 0.71 NISCH (0.69) NISCHADRA2BADRA2CADRA2A
SCHEMBL11428144 0.69 NISCH (0.55) NISCHADRA2BADRA2CADRA2AHTR1D
SCHEMBL8091334 0.69 NISCH (1.00) NISCHADRA2BADRA2CADRA2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4526897-A Hypertensive agents BEIERSDORF AKTIENGESELLSCHAFT (DE) 1985-07-02 US disclosed
EP-0072954-A2 Isoindolin-2-yl-amino-imidazolines and isoindolin-2-yl guanidines, process for their preparation and their use as medicines Beiersdorf Aktiengesellschaft (DE) 1983-03-02 EP disclosed