SCHEMBL11007474

SCHEMBL11007474

Brc1ccc(Br)c2c1CN(NC1=NCCN1)C2

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.58
ADRA2A P08913 10/20 0.42
ADRA2C P18825 8/20 0.42
ADRA2B P18089 7/20 0.42
ADRA1A P35348 2/20 0.39
CFB P00751 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
ADRA1D P25100 1/20 0.38
ADRA1B P35368 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10765153 0.92 NISCH (0.51) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL11007271 0.92 NISCH (0.51) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL10764582 0.81 NISCH (0.74) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL10767501 0.81 NISCH (0.58) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL10765612 0.77 NISCH (0.54) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL11003828 0.77 NISCH (0.54) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL6054462 0.77 NISCH (0.69) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL11006239 0.75 NISCH (0.52) NISCHADRA2AADRA2CADRA2BHTR1D
SCHEMBL11001474 0.74 NISCH (0.72) NISCHADRA2AADRA2CADRA2BADRA1A
SCHEMBL8091334 0.74 NISCH (1.00) NISCHADRA2AADRA2CADRA2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4526897-A Hypertensive agents BEIERSDORF AKTIENGESELLSCHAFT (DE) 1985-07-02 US disclosed
EP-0072954-A2 Isoindolin-2-yl-amino-imidazolines and isoindolin-2-yl guanidines, process for their preparation and their use as medicines Beiersdorf Aktiengesellschaft (DE) 1983-03-02 EP disclosed