SCHEMBL11008151

SCHEMBL11008151

CCOC(=O)C1=C(C)NC2=C(C(=O)OC2)C1c1ccccc1-c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.74
KDM4E B2RXH2 4/20 0.74
CACNA1C Q13936 2/20 0.49
NPSR1 Q6W5P4 3/20 0.49
MAPT P10636 3/20 0.49
GAA P10253 2/20 0.49
MGAM O43451 1/20 0.49
AMY1A P0DUB6 1/20 0.49
SI P14410 1/20 0.49
MGAM2 Q2M2H8 1/20 0.49
ADORA3 P0DMS8 2/20 0.47
CACNA1F O60840 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 1/20 0.44
AGTR1 P30556 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10730869 0.87 KDM4E (0.76) ALDH1A1KDM4ENPSR1MAPTGAA
SCHEMBL10659837 0.87 KDM4E (0.61) ALDH1A1KDM4ECACNA1CNPSR1MAPT
SCHEMBL9637750 0.86 KDM4E (0.74) ALDH1A1KDM4ENPSR1MAPTGAA
SCHEMBL11010941 0.86 KDM4E (0.74) ALDH1A1KDM4ENPSR1MAPTGAA
SCHEMBL9689623 0.86 ALDH1A1 (0.57) ALDH1A1KDM4ECACNA1CNPSR1MAPT
SCHEMBL7379319 0.85 ALDH1A1 (0.73) ALDH1A1KDM4ECACNA1CNPSR1MAPT
Hydrochloric Acid SCHEMBL10334321 0.85 KDM4E (0.73) ALDH1A1KDM4ENPSR1MAPTGAA
SCHEMBL11003495 0.85 KDM4E (0.69) ALDH1A1KDM4ECACNA1CCACNA1FCACNA1D
SCHEMBL7383959 0.84 KDM4E (0.72) ALDH1A1KDM4ENPSR1MAPTGAA
SCHEMBL11012267 0.84 KDM4E (0.68) ALDH1A1KDM4ECACNA1CNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed