SCHEMBL11010604

SCHEMBL11010604

CCCc1ccc(CO)c(CC)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
BACE1 P56817 1/20 0.46
VDR P11473 2/20 0.44
ALOX5 P09917 1/20 0.41
GPR84 Q9NQS5 3/20 0.40
LPL P06858 1/20 0.39
LIPG Q9Y5X9 1/20 0.39
PLK1 P53350 1/20 0.39
THRB P10828 1/20 0.38
CA2 P00918 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MCL1 Q07820 1/20 0.37
MTNR1A P48039 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13953779 0.92 CNR1 (0.50) CNR1CNR2BACE1VDRALOX5
SCHEMBL11720734 0.90 CNR1 (0.48) CNR1CNR2BACE1VDRALOX5
SCHEMBL9734907 0.87 CNR1 (0.48) CNR1CNR2BACE1ALOX5GPR84
SCHEMBL22490117 0.85 EGFR (0.46) BACE1VDRCA2
SCHEMBL606251 0.85 TRPA1 (0.46) BACE1LPLLIPGL3MBTL1
SCHEMBL28635844 0.85 TYR (0.50) CNR1CNR2VDRALOX5LPL
SCHEMBL14922851 0.84 BACE1 (0.42) CNR1CNR2BACE1VDRALOX5
SCHEMBL6756665 0.83 VDR (0.47) CNR1CNR2VDRALOX5LPL
SCHEMBL18007124 0.82 CNR1 (0.48) CNR1CNR2BACE1VDRALOX5
SCHEMBL11010600 0.82 CNR1 (0.44) CNR1CNR2BACE1ALOX5GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4537720-A N-substituted-2-(R)-(sulfinic acid)-3-(S)-(acylamino)-4-oxo-azetidines and process ELI LILLY AND COMPANY (US) 1985-08-27 US disclosed
US-4477660-A 7-(S)-Acylaminocephalosporin sulfones and process ELI LILLY AND COMPANY (US) 1984-10-16 US disclosed
US-4474879-A Process for 3-hydroxymethyl cephalosporin sulfones ELI LILLY AND COMPANY (US) 1984-10-02 US disclosed
US-4459405-A Desacetylcephalosporin sulfones ELI LILLY AND COMPANY (US) 1984-07-10 US disclosed
EP-0109301-A2 7-(S)-acylaminocephalosporin sulfones and process ELI LILLY AND COMPANY (US) 1984-05-23 EP disclosed
EP-0109300-A2 Desacetylcephalosporin sulfones ELI LILLY AND COMPANY (US) 1984-05-23 EP disclosed
US-4436596-A N-Substituted-2-(R)-(sulfinic acid)-3-(S)-(acylamido)-4-oxo-azetidines and process ELI LILLY AND COMPANY (US) 1984-03-13 US disclosed