SCHEMBL11020518

SCHEMBL11020518

COc1ccc(-c2nc(SCC(=O)N(C)C)nn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.51
PTGS1 P23219 4/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GAA P10253 1/20 0.44
ALOX5 P09917 2/20 0.43
MALT1 Q9UDY8 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
LIPE Q05469 1/20 0.43
TSPO P30536 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11019659 0.87 PTGS2 (0.54) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11040012 0.86 SMN1; SMN2 (0.56) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11021833 0.86 PTGS2 (0.53) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11051240 0.81 ALDH1A1 (0.55) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11053224 0.80 PTGS2 (0.57) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11022603 0.79 PTGS2 (0.56) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL6132198 0.78 PTGS2 (0.62) PTGS2PTGS1L3MBTL1KDM4EALDH1A1
SCHEMBL11021658 0.77 PTGS2 (0.53) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11020965 0.76 PTGS1 (0.56) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E
SCHEMBL11049382 0.76 PTGS2 (0.56) PTGS2PTGS1L3MBTL1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0157259-A1 3-Mercapto-1,2,4-triazacycloalcadiene derivatives CIBA-GEIGY AG (CH) 1985-10-09 EP claimed
EP-0157259-A1 3-Mercapto-1,2,4-triazacycloalcadiene derivatives CIBA-GEIGY AG (CH) 1985-10-09 EP disclosed