SCHEMBL11024331

SCHEMBL11024331

CCOC(=O)[C@@H]1Cc2ccc(N)cc2CN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
OPRM1 P35372 3/20 0.40
OPRD1 P41143 3/20 0.40
OPRK1 P41145 3/20 0.40
HDAC8 Q9BY41 8/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11028996 0.83 TSHR (0.44) OPRM1OPRD1OPRK1HDAC8MEN1
SCHEMBL31669038 0.82 KDM4E (0.57) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
SCHEMBL7744084 0.82 KDM4E (0.57) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
SCHEMBL3319088 0.82 KDM4E (0.57) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
SCHEMBL7743516 0.82 KDM4E (0.57) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
SCHEMBL16140165 0.81 TNF (0.41) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8121954 0.81 KDM4E (0.60) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8702078 0.81 KDM4E (0.60) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL30377815 0.81 KDM4E (0.60) KDM4EHSD17B10CYP1A2CYP2D6CYP2C9
SCHEMBL11030539 0.80 PNMT (0.62) ADRA2APNMTADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088350-B1 CARBOXYALKYL DIPEPTIDES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING CORPORATION (US) 1985-02-20 EP disclosed
EP-0088350-A1 Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them SCHERING CORPORATION (US) 1983-09-14 EP disclosed