SCHEMBL11024835

SCHEMBL11024835

Clc1ccc2[c]c3ccccc3[c]c2c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.44
TP53 P04637 2/20 0.38
S100A4 P26447 1/20 0.37
TSHR P16473 7/20 0.36
CYP1A2 P05177 1/20 0.36
AHR P35869 2/20 0.35
GPR3 P46089 1/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 4/20 0.35
ALDH1A1 P00352 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALOX15 P16050 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PNMT P11086 1/20 0.34
HSD17B10 Q99714 3/20 0.33
MEN1 O00255 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11030089 0.92 TP53 (0.43) CYP2A6TP53S100A4TSHRAHR
SCHEMBL11025889 0.78 CYP3A4 (0.37) CYP2A6TP53CYP1A2LMNACYP3A4
SCHEMBL11028225 0.78 CYP3A4 (0.37) CYP2A6TP53CYP1A2LMNACYP3A4
SCHEMBL70153 0.76 CYP2A6 (0.36) CYP2A6TSHRLMNACYP3A4ALDH1A1
SCHEMBL508847 0.72 CYP2A6 (0.39) CYP2A6TP53TSHRCYP1A2CYP3A4
SCHEMBL1263751 0.72 TDP1 (0.42) CYP2A6TP53TSHRCYP1A2LMNA
SCHEMBL2022581 0.70 MAOA (0.44) CYP1A2LMNACYP3A4ALDH1A1TDP1
SCHEMBL509988 0.68 ALDH1A1 (0.42) CYP2A6TP53TSHRCYP1A2CYP3A4
SCHEMBL2025646 0.67 ALDH1A1 (0.42) TSHRCYP1A2LMNAALDH1A1TDP1
SCHEMBL508867 0.65 CYP2A6 (0.44) CYP2A6TP53TSHRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0053937-B1 POLYNUCLEAR FUSED AROMATIC RING TYPE POLYMER AND PREPARATION THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1985-06-19 EP claimed
US-4463162-A POLYESTERS FROM ANTHRACENEDIOL ASAHI-DOW LIMITED (JP) 1984-07-31 US claimed
EP-0053937-A1 Polynuclear fused aromatic ring type polymer and preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-06-16 EP claimed
EP-0053937-B1 POLYNUCLEAR FUSED AROMATIC RING TYPE POLYMER AND PREPARATION THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1985-06-19 EP disclosed
US-4463162-A POLYESTERS FROM ANTHRACENEDIOL ASAHI-DOW LIMITED (JP) 1984-07-31 US disclosed
EP-0053937-A1 Polynuclear fused aromatic ring type polymer and preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-06-16 EP disclosed