SCHEMBL11026470

SCHEMBL11026470

CC(C)(CO)CNc1nc(N2CC[S+]([O-])CC2)c2ncnc(SCc3ccccc3)c2n1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 16/20 0.36
CYP1A2 P05177 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
PPARG P37231 1/20 0.35
NCOA2 Q15596 1/20 0.35
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11049468 0.88 NPSR1 (0.38) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL2460092 0.87 SLC29A1 (0.45) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL10970925 0.86 SLC29A1 (0.43) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL10969544 0.86 ALDH1A1 (0.41) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL10969508 0.85 SLC29A1 (0.38) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL11046570 0.85 CYP1A2 (0.40) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL11050061 0.85 CYP1A2 (0.38) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL11026335 0.84 PDE4A (0.44) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL10971507 0.84 CYP1A2 (0.37) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9
SCHEMBL11049547 0.84 SLC29A1 (0.40) SLC29A1CYP1A2KDM4EALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055444-B1 TRISUBSTITUTED PYRIMIDO(5,4-D)PYRIMIDINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-03-20 EP disclosed
US-4478833-A ANTICOAGULANTS DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-10-23 US disclosed
EP-0055444-A2 Trisubstituted pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-07-07 EP disclosed