SCHEMBL11029941

SCHEMBL11029941

O=[N+]([O-])c1cccc(OCC(F)(F)F)c1OCC(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
RECQL P46063 2/20 0.51
ALDH1A1 P00352 6/20 0.46
HSPB1 P04792 1/20 0.46
HTT P42858 1/20 0.46
POLB P06746 1/20 0.44
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 3/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CFTR P13569 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11451550 0.90 RECQL (0.49) NPC1RAB9ARECQLALDH1A1HSPB1
SCHEMBL31194220 0.89 RAB9A (0.66) NPC1RAB9ARECQLALDH1A1HTT
SCHEMBL4185071 0.89 RAB9A (0.66) NPC1RAB9ARECQLALDH1A1HTT
SCHEMBL28345439 0.84 HSPB1 (0.46) NPC1RAB9ARECQLALDH1A1HSPB1
SCHEMBL28504880 0.84 NPC1 (0.47) NPC1RAB9ARECQLALDH1A1HSPB1
SCHEMBL10532607 0.83 MAPT (0.44) NPC1RAB9ARECQLALDH1A1POLB
SCHEMBL28649512 0.83 NPC1 (0.42) NPC1RAB9ARECQLALDH1A1HSPB1
SCHEMBL27585308 0.80 TDP1 (0.50) NPC1RAB9ARECQLALDH1A1HTT
SCHEMBL17276070 0.79 NPC1 (0.56) NPC1RAB9ARECQLALDH1A1HSPB1
SCHEMBL29740003 0.79 P2RX1 (0.45) NPC1RAB9ARECQLALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4491584-A ANTIARRHYTHMIA AGENTS RIKER LABORATORIES (US) 1985-01-01 US disclosed
US-4154941-A ANTIARRHYTHMIC AGENTS RIKER LABORATORIES, INC. (US) 1979-05-15 US disclosed
US-4071524-A Derivatives of urea RIKER LABORATORIES, INC. (US) 1978-01-31 US disclosed