SCHEMBL110311

SCHEMBL110311

C[Si](C)(C)CCOCn1cnc2cc(N3CCC(NC(=O)O)C3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 9/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
KLKB1 P03952 1/20 0.36
DGAT1 O75907 1/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
USP2 O75604 1/20 0.35
RAB9A P51151 1/20 0.35
MAPK1 P28482 1/20 0.34
MAPT P10636 2/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
CACNA2D1 P54289 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2129492 0.89 SUV39H2 (0.41)
SCHEMBL2143659 0.83 MET (0.41)
SCHEMBL108873 0.80 PTGDR (0.37) DGAT1
SCHEMBL2142224 0.78 CCNE1 (0.37) DGAT1
SCHEMBL31540053 0.76 NTRK1 (0.38) DGAT1ALDH1A1NPC1
SCHEMBL2143614 0.76 NTRK1 (0.46) DGAT1ALDH1A1NPC1RAB9AMAPK1
SCHEMBL26124012 0.75 DGAT1 (0.36) MTNR1AMTNR1BKLKB1DGAT1CACNA2D1
SCHEMBL2128838 0.74 MAPT (0.43) ALDH1A1MAPT
SCHEMBL25426997 0.73 GNRHR (0.43) ALDH1A1NPC1USP2RAB9AMAPT
SCHEMBL30508603 0.73 GNRHR (0.43) ALDH1A1NPC1USP2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424843-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES Novartis AG (CH) 2012-03-07 EP disclosed
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed