SCHEMBL11032483

SCHEMBL11032483

NC(Cn1ccc2cc(F)ccc21)C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 11/20 0.65
HTR2A P28223 9/20 0.65
PRMT5 O14744 1/20 0.46
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CYP1A2 P05177 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GRIA1 P42261 1/20 0.42
GRIA2 P42262 1/20 0.42
GRIA3 P42263 1/20 0.42
GRIA4 P48058 1/20 0.42
GRIK5 Q16478 1/20 0.42
P2RX7 Q99572 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042962 0.83 HTR2C (0.65) HTR2CHTR2APRMT5HDAC3HDAC1
SCHEMBL4042963 0.83 HTR2C (0.65) HTR2CHTR2APRMT5HDAC3HDAC1
SCHEMBL11033586 0.81 HTR2C (0.68) HTR2CHTR2APRMT5HDAC8HDAC6
Fumaric Acid SCHEMBL8959477 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
Fumaric Acid SCHEMBL8959680 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
Fumaric Acid SCHEMBL8959800 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
Fumaric Acid SCHEMBL8959669 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
Fumaric Acid SCHEMBL8959482 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
Fumaric Acid SCHEMBL8959795 0.80 HTR2C (0.78) HTR2CHTR2APRMT5CYP1A2CYP3A4
SCHEMBL8191415 0.79 KMT2A (0.58) HDAC1HDAC2HDAC8HDAC6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448785-A N-Unsaturated fatty acid amides of tryptophan ester homologues and anti-cholesteric use thereof SANDOZ, INC. (US) 1984-05-15 US disclosed