SCHEMBL11034855

SCHEMBL11034855

C=CCn1c(=O)c2[nH]c3nc2n(o3)c1=O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.46
ADORA2A P29274 4/20 0.46
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
ADORA3 P0DMS8 2/20 0.40
ADORA1 P30542 1/20 0.40
CYP3A4 P08684 2/20 0.38
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9122677 0.71 ADORA2B (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL18127922 0.71 ADORA2B (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL7112265 0.70 ADORA2B (0.54) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL11029795 0.69 ADORA2B (0.46) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10856290 0.67 ADORA2B (0.61) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL27473174 0.66 ADORA2B (0.43) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL3435824 0.65 ADORA2B (0.80) ADORA2BADORA2AADORA3ADORA1CYP3A4
SCHEMBL4953015 0.65 ADORA2B (0.52) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10857602 0.65 PDE1A (0.66) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10629155 0.65 ADORA1 (0.67) ADORA2BADORA2AADORA3ADORA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed