SCHEMBL11029795

SCHEMBL11029795

C=CCn1c(=O)c2[nH]c(O)nc2n(O)c1=O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.46
ADORA2A P29274 4/20 0.46
ADORA3 P0DMS8 2/20 0.42
ADORA1 P30542 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
CYP3A4 P08684 1/20 0.38
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5404111 0.81 SIRT1 (0.51) ADORA2BADORA2AADORA3ADORA1PDE4A
SCHEMBL11033010 0.75 ADORA2B (0.48) ADORA2BADORA2AADORA1PDE4APDE4B
SCHEMBL27471745 0.74 ADORA2B (0.57) ADORA2BADORA2AADORA3ADORA1CYP3A4
SCHEMBL18127922 0.71 ADORA2B (0.55) ADORA2BADORA2AADORA3ADORA1PDE4A
SCHEMBL9122677 0.71 ADORA2B (0.55) ADORA2BADORA2AADORA3ADORA1PDE4A
SCHEMBL7112265 0.70 ADORA2B (0.54) ADORA2BADORA2AADORA3ADORA1PDE4A
SCHEMBL10747983 0.69 ADORA2B (0.70) ADORA2BADORA2AADORA3ADORA1CYP3A4
SCHEMBL11044972 0.69 ADORA2B (0.42) ADORA2BADORA2AADORA3ADORA1CYP3A4
SCHEMBL21393356 0.69 MEN1 (0.56) ADORA2BADORA2ACYP3A4LMNAUSP2
SCHEMBL11034855 0.69 ADORA2B (0.46) ADORA2BADORA2AADORA3ADORA1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed