SCHEMBL11035104

SCHEMBL11035104

Nc1ncc([N+](=O)[O-])c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.50
CTSB P07858 4/20 0.49
ALDH1A1 P00352 6/20 0.44
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
POLB P06746 1/20 0.42
HPRT1 P00492 1/20 0.42
MAPT P10636 4/20 0.41
PIN1 Q13526 2/20 0.41
KDM4E B2RXH2 4/20 0.40
CYP3A4 P08684 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GSK3B P49841 1/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21437204 0.81 MAPT (0.48) TDP1ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL9836130 0.79 TDP1 (0.62) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL2431427 0.78 TDP1 (0.50) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL12314708 0.78 TDP1 (0.50) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL4470384 0.78 CTSB (0.55) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL29532198 0.78 TDP1 (0.50) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL27995682 0.78 TDP1 (0.50) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL202880 0.75 POLB (0.51) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL14089776 0.74 CTSB (0.46) TDP1CTSBALDH1A1NCOA1NCOA3
SCHEMBL27006369 0.74 PIN1 (0.49) TDP1CTSBALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-59172472-A None JP disclosed
CN-101296924-A Pyrazole-isoquinoline urea derivatives as P38 kinase inhibitors LILLY CO ELI (US) 2008-10-29 CN disclosed
JP-S59172472-A ISOQUINOLINE DERIVATIVE AND ITS SALT, THEIR PREPARATION, AND ANTIALLERGIC AGENT CONTAINING SAID COMPOUND AS ACTIVE COMPONENT FUJISAWA PHARMACEUT CO LTD 1984-09-29 JP disclosed