SCHEMBL11039239

SCHEMBL11039239

[CH2]COc1cccc2c1OCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.41
MTNR1A P48039 4/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AOC3 Q16853 1/20 0.37
EED O75530 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR2A P28223 2/20 0.35
HTR2C P28335 1/20 0.35
GSK3B P49841 1/20 0.35
TTBK1 Q5TCY1 1/20 0.35
TTBK2 Q6IQ55 1/20 0.35
MGAM O43451 1/20 0.35
AMY1A P0DUB6 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236657 0.86 MTNR1A (0.54) HTR1AMTNR1A
SCHEMBL13534203 0.82 AOC3 (0.54) HTR1AMTNR1AABCG2KMT2AAOC3
SCHEMBL27443068 0.81 ALDH1A1 (0.45) HTR1AMTNR1AKMT2ATDP1L3MBTL1
SCHEMBL1145696 0.79 ABCG2 (0.44) HTR1AMTNR1AABCG2KMT2ATDP1
SCHEMBL4309152 0.79 MTNR1A (0.48) HTR1AMTNR1AABCG2KMT2ATDP1
SCHEMBL9239494 0.79 MTNR1A (0.47) HTR1AMTNR1AABCG2KMT2ATDP1
SCHEMBL25335293 0.78 HTR1B (0.46) HTR1AMTNR1AABCG2KMT2ATDP1
SCHEMBL13533388 0.78 TP53 (0.44) HTR1AMTNR1AABCG2KMT2ATDP1
SCHEMBL13534270 0.78 MTNR1A (0.50) HTR1AMTNR1AKMT2ATDP1L3MBTL1
SCHEMBL17274865 0.78 MAPT (0.44) HTR1AMTNR1AABCG2KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed