SCHEMBL11040283

SCHEMBL11040283

CCOc1ccc(F)cc1C1OC(=O)NC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.47
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
HTR2A P28223 1/20 0.38
MAPK1 P28482 1/20 0.38
PPARG P37231 7/20 0.37
PPARD Q03181 2/20 0.37
PPARA Q07869 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11041960 0.85 CA2 (0.60) CA2HTR2CHTR2BHTR2A
SCHEMBL11040416 0.84 HTR2C (0.48) CA2HTR2CHTR2BHTR2APPARG
SCHEMBL11040310 0.83 CA2 (0.51) CA2HTR2CHTR2BHTR2AMAPK1
SCHEMBL11038153 0.78 CA2 (0.43) CA2PPARGPPARDPPARAKDM4E
SCHEMBL10547400 0.78 CA2 (0.40) CA2PPARGPPARDPPARA
SCHEMBL11040694 0.77 CA2 (0.47) CA2LMNAPDE3BPDE3AKDM4E
SCHEMBL10892219 0.74 CA2 (0.44) CA2PPARGPPARDPPARALMNA
SCHEMBL11044359 0.70 CA2 (0.43) CA2MAPK1PPARGPPARDPPARA
SCHEMBL21816496 0.70 SLC6A2 (0.48) HTR2CHTR2BHTR2A
SCHEMBL11043516 0.70 CA2 (0.62) CA2MAPK1SMN1; SMN2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448971-A Hypoglycemic 5-phenyl-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1984-05-15 US disclosed
US-4407811-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-10-04 US disclosed
US-4399296-A TRIMETHYLSILYL CYANOHYDRIN INTERMEDIATES PFIZER INC. (US) 1983-08-16 US disclosed
US-4367234-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1983-01-04 US disclosed