SCHEMBL11043337

SCHEMBL11043337

CC(=O)Nc1ccc(C(=O)CCN2CCN(C(=O)c3ccc4c(c3)CCC(=O)N4)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.49
HTR2A P28223 3/20 0.49
HTR7 P34969 3/20 0.49
DRD3 P35462 3/20 0.49
DRD4 P21917 2/20 0.49
NR3C1 P04150 1/20 0.48
PGR P06401 1/20 0.48
SLC6A4 P31645 1/20 0.48
KCNH2 Q12809 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
CRBN Q96SW2 6/20 0.46
CYP2C19 P33261 1/20 0.43
SMYD3 Q9H7B4 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ROCK2 O75116 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044792 0.87 NR3C1 (0.52) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL7294275 0.86 KMT2A (0.58) HTR1AHTR2AHTR7DRD3DRD4
Hydrochloric Acid SCHEMBL11041436 0.85 KMT2A (0.57) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL7286669 0.85 HTR1A (0.51) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL7325459 0.85 NR3C1 (0.56) HTR1AHTR2AHTR7DRD3DRD4
Hydrochloric Acid SCHEMBL7295612 0.83 KMT2A (0.51) HTR1AHTR2AHTR7DRD3DRD4
Hydrochloric Acid SCHEMBL11043902 0.83 KMT2A (0.55) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL11046347 0.79 NR3C1 (0.62) NR3C1PGRSLC6A4KCNH2PDE3B
Water SCHEMBL11039451 0.78 NR3C1 (0.54) HTR1AHTR2AHTR7DRD3DRD4
Iodide SCHEMBL11041065 0.78 NR3C1 (0.61) NR3C1PGRSLC6A4KCNH2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed