SCHEMBL11044017

SCHEMBL11044017

C/C(=C\c1ccccc1)C(=O)c1ccccc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.58
MAPT P10636 5/20 0.50
BCHE P06276 1/20 0.50
DHODH Q02127 1/20 0.50
TRPM8 Q7Z2W7 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
HPGD P15428 3/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
HMGB1 P09429 1/20 0.48
CA4 P22748 1/20 0.48
CA6 P23280 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
NAPRT Q6XQN6 1/20 0.48
CA14 Q9ULX7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044018 1.00 AKR1C3 (0.58) AKR1C3MAPTBCHEDHODHTRPM8
SCHEMBL1073512 0.83 MAPT (0.55) AKR1C3MAPTBCHECYP2C19ALDH1A1
SCHEMBL4865622 0.82 AKR1C3 (0.58) AKR1C3MAPTDHODHTRPM8ALDH1A1
SCHEMBL11561505 0.79 MAPT (0.50) MAPTBCHECYP2C19ALDH1A1KDM4E
SCHEMBL1649381 0.79 MAPT (0.50) AKR1C3MAPTBCHECYP2C19ALDH1A1
SCHEMBL4050625 0.79 MAPT (0.50) AKR1C3MAPTBCHECYP2C19ALDH1A1
SCHEMBL11561504 0.79 MAPT (0.50) MAPTBCHECYP2C19ALDH1A1KDM4E
SCHEMBL27977683 0.77 AKR1C1 (0.59) AKR1C3MAPTBCHECYP2C19ALDH1A1
SCHEMBL30495367 0.77 MAPT (0.47) AKR1C3MAPTBCHEDHODHTRPM8
SCHEMBL11203024 0.77 MAPT (0.47) AKR1C3MAPTBCHEDHODHTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025599-B1 BENZOPYRAN COMPOUNDS, USEFUL AS CHEMOTHERAPEUTIC AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1984-12-19 EP disclosed
US-4452991-A OR BENZO(B)INDENO (2,1-E) PYRANS OR BENZO(C)XANTHENES BATCHELOR JOHN F (GB) 1984-06-05 US disclosed
EP-0025599-A1 Benzopyran compounds, useful as chemotherapeutic agents THE WELLCOME FOUNDATION LIMITED (GB) 1981-03-25 EP disclosed