SCHEMBL11044555

SCHEMBL11044555

Cc1ccc(C(=O)N2CCN(C(=O)c3ccc4c(c3)CCC(=O)N4)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.60
NR3C1 P04150 1/20 0.60
PGR P06401 1/20 0.60
SLC6A4 P31645 1/20 0.60
PDE3B Q13370 1/20 0.60
PDE3A Q14432 1/20 0.60
CRBN Q96SW2 6/20 0.57
PKM P14618 3/20 0.52
ALDH1A1 P00352 2/20 0.50
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47
GABRA4 P48169 1/20 0.47
HPGD P15428 1/20 0.47
OGT O15294 1/20 0.46
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341674 0.90 ALDH1A1 (0.53) KCNH2NR3C1PGRSLC6A4PDE3B
SCHEMBL11046347 0.90 NR3C1 (0.62) KCNH2NR3C1PGRSLC6A4PDE3B
Hydrochloric Acid SCHEMBL11044714 0.89 NR3C1 (0.52) KCNH2NR3C1PGRSLC6A4PDE3B
Hydrochloric Acid SCHEMBL11041427 0.89 NR3C1 (0.52) KCNH2NR3C1PGRSLC6A4PDE3B
Iodide SCHEMBL11041065 0.88 NR3C1 (0.61) KCNH2NR3C1PGRSLC6A4PDE3B
Hydrochloric Acid SCHEMBL7348598 0.88 ALDH1A1 (0.51) KCNH2NR3C1PGRSLC6A4PDE3B
SCHEMBL11042243 0.88 ALDH1A1 (0.61) KCNH2NR3C1PGRSLC6A4PDE3B
SCHEMBL11044792 0.88 NR3C1 (0.52) KCNH2NR3C1PGRSLC6A4PDE3B
SCHEMBL11044078 0.87 NR3C1 (0.57) KCNH2NR3C1PGRSLC6A4PDE3B
SCHEMBL11045054 0.87 CRBN (0.62) KCNH2NR3C1PGRSLC6A4PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed