SCHEMBL11045209

SCHEMBL11045209

CCOc1cccc(/C=C/[C]=O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.61
ALDH1A1 P00352 2/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
TLR4 O00206 1/20 0.47
TLR2 O60603 1/20 0.47
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
RELA Q04206 2/20 0.45
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
HDAC4 P56524 1/20 0.43
MEF2D Q14814 1/20 0.43
CCNB2 O95067 2/20 0.42
CDK1 P06493 2/20 0.42
CDK4 P11802 2/20 0.42
CCNB1 P14635 2/20 0.42
CCND1 P24385 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
MAOA P21397 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11045213 1.00 KDM4E (0.61) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL11041123 0.88 TLR4 (0.55) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL11041121 0.88 TLR4 (0.55) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL4414011 0.84 KDM4E (0.47) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL4414013 0.84 KDM4E (0.47) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL21457214 0.84 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL21457217 0.84 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL11045237 0.84 TLR4 (0.58) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL11045240 0.84 TLR4 (0.58) KDM4EALDH1A1SMN1; SMN2TLR4TLR2
SCHEMBL7342257 0.83 ESR1 (0.49) KDM4EALDH1A1SMN1; SMN2RELACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed