SCHEMBL11045809

SCHEMBL11045809

CC(C)(C)OC(=O)NC(F)(F)CF

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
CA12 O43570 2/20 0.36
CA14 Q9ULX7 2/20 0.36
CTSK P43235 5/20 0.35
DGAT1 O75907 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CYP2D6 P10635 1/20 0.34
AAK1 Q2M2I8 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13690847 0.81 APLNR (0.41) APLNRTDP1CA1CA2CA7
SCHEMBL28918296 0.78 APLNR (0.40) APLNRTDP1CA1CA2CA7
SCHEMBL2279581 0.76 MEN1 (0.39) APLNRTDP1CA1CA2CA7
SCHEMBL28682013 0.76 DGAT1 (0.45) APLNRTDP1CA1CA2CA7
SCHEMBL28672286 0.76 MEN1 (0.39) APLNRTDP1CA1CA2CA7
SCHEMBL5007482 0.76 MEN1 (0.39) APLNRTDP1CA1CA2CA7
SCHEMBL7279185 0.76 MEN1 (0.39) APLNRTDP1CA1CA2CA7
SCHEMBL2274474 0.76 DGAT1 (0.41) APLNRTDP1CA1CA2CA7
SCHEMBL28682014 0.76 DGAT1 (0.45) APLNRTDP1CA1CA2CA7
SCHEMBL8353864 0.74 APLNR (0.38) APLNRTDP1CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0098457-A2 (1S,2R,3R)- and (1R,2S,3S)-nitrilo-1-carbonyl-3-methyl-2-oxy-heptanes and -hept-5-enes useful in the total synthesis of cyclosporins and processes for their production SANDOZ AG (CH) 1984-01-18 EP disclosed
EP-0098456-A2 Peptides comprising a (1S,2R,3R)- or (1R,2S,3S)-1-nitrilo-1-carbonyl-3-methyl-2-oxy-heptane or -hept-5-ene residue useful in the total synthesis of cyclosporins, and processes for their production SANDOZ AG (CH) 1984-01-18 EP disclosed
EP-0034567-A2 A method for the total synthesis of cyclosporins and novel cyclosporins SANDOZ AG (CH) 1981-08-26 EP disclosed