SCHEMBL11049587

SCHEMBL11049587

c1cn(CCCC2CCCCCCC2)cn1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.64
HRH4 Q9H3N8 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
TBXAS1 P24557 9/20 0.55
GAA P10253 1/20 0.51
QPCT Q16769 1/20 0.51
CYP19A1 P11511 5/20 0.48
ALOX15 P16050 1/20 0.43
PRKCI P41743 1/20 0.42
TPSAB1 Q15661 1/20 0.42
TPSD1 Q9BZJ3 1/20 0.42
TPSG1 Q9NRR2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24833975 1.00 CYP2B6 (0.64) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL11047220 0.98 CYP2B6 (0.61) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL16163635 0.95 CYP2B6 (0.62) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL11051486 0.89 CYP2B6 (0.68) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL11050188 0.89 CYP2B6 (0.68) CYP2B6HRH4HRH3TBXAS1GAA
Iodide SCHEMBL16164357 0.88 CYP2B6 (0.66) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL24833961 0.87 CYP2B6 (0.53) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL10784468 0.84 TBXAS1 (0.49) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL11720830 0.84 TBXAS1 (0.53) CYP2B6HRH4HRH3TBXAS1GAA
SCHEMBL6174188 0.83 TBXAS1 (0.52) CYP2B6HRH4HRH3TBXAS1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4284641-A ANTITHROMBOEMBOLIC AGENT BURROUGHS WELLCOME CO. (US) 1981-08-18 US claimed
US-11571686-B2 Removal of homogeneous catalysts from NMR/MRI agents hyperpolarized via sabre or PHIP BOARD OF TRUSTEES OF SOUTHERN ILLINOIS UNIVERSITY (US) 2023-02-07 US disclosed
US-20230001400-A9 REMOVAL OF HOMOGENEOUS CATALYSTS FROM NMR/MRI AGENTS HYPERPOLARIZED VIA SABRE OR PHIP BOARD OF TRUSTEES OF SOUTHERN ILLINOIS UNIVERSITY (US) 2023-01-05 US disclosed
US-20210252493-A1 REMOVAL OF HOMOGENEOUS CATALYSTS FROM NMR/MRI AGENTS HYPERPOLARIZED VIA SABRE OR PHIP BOARD OF TRUSTEES OF SOUTHERN ILLINOIS UNIVERSITY (US) 2021-08-19 US disclosed
US-9556218-B2 Process for the preparation of abiraterone and intermediates thereof SCINOPHARM TAIWAN, LTD. (TW) 2017-01-31 US disclosed
EP-0000951-B1 PHARMACEUTICAL FORMULATIONS COMPRISING 1-SUBSTITUTED IMIDAZOLES, 1-SUBSTITUTED IMIDAZOLES AND 1-SUBSTITUTED IMIDAZOLES FOR USE IN THE TREATMENT OR PROPHYLAXIS OF THROMBO-EMBOLIC DISORDERS THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-23 EP disclosed
EP-0000950-B1 IMIDAZOLE DERIVATIVES AND SALTS THEREOF AND THEIR SYNTHESIS THE WELLCOME FOUNDATION LIMITED (GB) 1984-02-01 EP disclosed
US-4317830-A ANTISHOCK AGENTS, ANTICOAGULANTS BURROUGHS WELLCOME CO. (US) 1982-03-02 US disclosed
US-4284641-A ANTITHROMBOEMBOLIC AGENT BURROUGHS WELLCOME CO. (US) 1981-08-18 US disclosed
EP-0000950-A1 Imidazole derivatives and salts thereof and their synthesis THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP disclosed
EP-0000951-A1 Pharmaceutical Formulations comprising 1-substituted imidazoles, 1-substituted imidazoles and 1-substituted imidazoles for use in the treatment or prophylaxis of thrombo-embolic disorders THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP disclosed