SCHEMBL11047768

SCHEMBL11047768

COc1ccc2c(c1)CCC(C(=O)ON(C1CCCCC1)C1CCCCC1)N2C(=O)CCS

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.38
HSD17B10 Q99714 1/20 0.37
NOTUM Q6P988 1/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
MAPK1 P28482 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052936 0.84 ACE (0.42)
SCHEMBL11047749 0.82 ACE (0.45) MTNR1AHSD17B10NOTUMALDH1A1LMNA
SCHEMBL11046009 0.76 MEN1 (0.36) NOTUMALDH1A1LMNATSHRHTT
SCHEMBL11047662 0.76 ACE (0.43) MEN1KMT2A
SCHEMBL10921170 0.73 ACE (0.43)
SCHEMBL11051574 0.73 OPRL1 (0.40)
SCHEMBL11052123 0.71 MEN1 (0.32) LMNAHDAC1HDAC6MEN1NPC1
SCHEMBL7338202 0.70 NOTUM (0.48) MTNR1AHSD17B10NOTUMALDH1A1LMNA
SCHEMBL7336655 0.70 NOTUM (0.48) MTNR1AHSD17B10NOTUMALDH1A1LMNA
SCHEMBL7343636 0.70 NOTUM (0.48) MTNR1AHSD17B10NOTUMALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4461896-A 1-[Acylthio) and (mercapto)-1-oxoalkyl]-1,2,3,4-tetrahydroquinoline-2-carboxylic acids NORWICH EATON PHARMACEUTICALS, INC. (US) 1984-07-24 US disclosed