SCHEMBL11049752

SCHEMBL11049752

O=C1CCc2ccncc2C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
CYP11B1 P15538 6/20 0.50
CYP11B2 P19099 6/20 0.50
CYP1A2 P05177 5/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
CHRNB2 P17787 3/20 0.48
CHRNA4 P43681 3/20 0.48
PDE3B Q13370 3/20 0.33
PDE3A Q14432 3/20 0.33
DAO P14920 1/20 0.33
TIPARP Q7Z3E1 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP19A1 P11511 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
FDPS P14324 1/20 0.32
CHRNA7 P36544 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21899911 0.92 CYP11B1 (0.54) CYP2A6SIGMAR1CYP11B1CYP11B2CYP1A2
SCHEMBL12797257 0.88 SIGMAR1 (0.61) CYP2A6SIGMAR1CYP11B1CYP11B2CYP1A2
SCHEMBL7343370 0.85 CYP1A2 (0.50) CYP2A6SIGMAR1CYP11B1CYP11B2CYP1A2
SCHEMBL11265173 0.80 SIGMAR1 (0.61) CYP2A6SIGMAR1CYP11B1CYP11B2CYP1A2
SCHEMBL8348679 0.79
SCHEMBL8419080 0.74 SIGMAR1 (0.56) CYP2A6SIGMAR1CYP1A2CYP3A4CYP2C9
SCHEMBL20682524 0.73 SIGMAR1 (0.95) SIGMAR1CYP11B1CYP11B2CHRNB2CHRNA4
Ammonia Solution, Strong SCHEMBL28923744 0.72
5,6,7,8-Tetrahydroisoquinoline SCHEMBL28211 0.70 SIGMAR1 (1.00) SIGMAR1CYP11B1CYP11B2CHRNB2CHRNA4
SCHEMBL29518090 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114133389-B Process for preparing isoindolin-1-one fused rings and analogues thereof 海南梵圣生物科技有限公司 2023-03-21 CN disclosed
CN-114133389-A Process for preparing isoindolin-1-one fused rings and analogues thereof 海南梵圣生物科技有限公司 2022-03-04 CN disclosed
US-4468400-A PEPTIC ULCERS SCHERING CORPORATION (US) 1984-08-28 US disclosed