SCHEMBL11050220

SCHEMBL11050220

COCCNc1ncn(-c2c(C)cccc2Cl)c(=O)n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
MAPK14 Q16539 1/20 0.41
CHRNA7 P36544 14/20 0.41
HSD17B10 Q99714 2/20 0.39
HTT P42858 1/20 0.39
EGFR P00533 1/20 0.37
FGFR1 P11362 1/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056120 0.89 MKNK1 (0.43) SMN1; SMN2ALDH1A1KDM4EMKNK1MKNK2
SCHEMBL11056350 0.88 MKNK1 (0.43) SMN1; SMN2ALDH1A1KDM4EMKNK1MKNK2
SCHEMBL11050309 0.87 CHRNA7 (0.43) MAPK14CHRNA7EGFRFGFR1
SCHEMBL11053108 0.87 MKNK1 (0.43) SMN1; SMN2ALDH1A1KDM4EMKNK1MKNK2
SCHEMBL11059310 0.86 CHRNA7 (0.44) MAPK14CHRNA7FGFR1
SCHEMBL11058225 0.85 EGFR (0.46) CHRNA7EGFRFGFR1
SCHEMBL11058286 0.85 EGFR (0.45) ALDH1A1CHRNA7HSD17B10EGFRFGFR1
SCHEMBL11055055 0.85 CHRNA7 (0.43) MKNK2MAPK14CHRNA7FGFR1
SCHEMBL11060182 0.83 CHRNA7 (0.43) CHRNA7EGFRFGFR1
SCHEMBL11052662 0.82 MKNK1 (0.49) SMN1; SMN2ALDH1A1KDM4EMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed