SCHEMBL11050274

SCHEMBL11050274

CC(=O)Oc1ccc([C@H]2CC(=O)c3cc(OC(C)=O)cc(OC(C)=O)c3O2)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.51
ABCG2 Q9UNQ0 2/20 0.47
ABCB1 P08183 1/20 0.47
AR P10275 1/20 0.47
ACHE P22303 3/20 0.47
BCHE P06276 2/20 0.47
MAOB P27338 5/20 0.45
CYP19A1 P11511 3/20 0.45
CYP3A4 P08684 1/20 0.45
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11641394 0.91 CYP3A4 (0.50) PTPN1CYP19A1CYP3A4NPC1RAB9A
SCHEMBL2399205 0.86 SLC22A12 (0.50) PTPN1ABCG2ABCB1ARACHE
SCHEMBL29477373 0.81 BCHE (0.69) ABCG2ACHEBCHECYP19A1CYP3A4
SCHEMBL31022637 0.81 BCHE (0.69) ABCG2ACHEBCHECYP19A1CYP3A4
SCHEMBL6726363 0.81 BCHE (0.69) ABCG2ACHEBCHECYP19A1CYP3A4
SCHEMBL6726368 0.81 BCHE (0.69) ABCG2ACHEBCHECYP19A1CYP3A4
SCHEMBL2399200 0.79 MAOB (0.68) MAOBCYP19A1CYP3A4
SCHEMBL17138198 0.78 GAA (0.45) ABCG2ABCB1ARACHEBCHE
SCHEMBL6723899 0.78 MAOB (0.62) ABCG2ABCB1ARACHEMAOB
SCHEMBL11636342 0.77 CYP19A1 (0.50) PTPN1ABCG2ABCB1ARACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4461907-A Amino-substituted flavans useful as anti-viral agents BURROUGHS WELLCOME CO. 1984-07-24 US disclosed
EP-0004579-B1 FLAVANS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1982-08-18 EP disclosed
EP-0051061-A2 Novel intermediates and process for their preparation THE WELLCOME FOUNDATION LIMITED (GB) 1982-05-05 EP disclosed
EP-0004579-A1 Flavans, process for their preparation and pharmaceutical compositions containing them THE WELLCOME FOUNDATION LIMITED (GB) 1979-10-17 EP disclosed