SCHEMBL11053485

SCHEMBL11053485

CCc1cc(O)cc(CC)c1-n1cnc(NC)nc1=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 10/20 0.41
ESR1 P03372 9/20 0.41
AURKA O14965 1/20 0.31
HPGD P15428 2/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30
LCK P06239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11059249 0.92 ESR1 (0.38) ESR2ESR1LCK
SCHEMBL11055393 0.91 ESR1 (0.38) ESR2ESR1
SCHEMBL11052642 0.91 ESR1 (0.38) ESR2ESR1
SCHEMBL11055572 0.91 ESR1 (0.38) ESR2ESR1
SCHEMBL11474313 0.87 MEN1 (0.31) LMNA
SCHEMBL11053551 0.87 ESR1 (0.34) ESR2ESR1
SCHEMBL11354153 0.86 EGFR (0.36)
SCHEMBL11344723 0.86 NPC1 (0.32)
SCHEMBL11058852 0.86 ELANE (0.34) AURKA
SCHEMBL11498090 0.85 ESR1 (0.34) ESR2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed