SCHEMBL11059249

SCHEMBL11059249

CCc1cc(O)cc(C)c1-n1cnc(NC)nc1=O

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.38
ESR2 Q92731 8/20 0.38
WEE1 P30291 1/20 0.30
LCK P06239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053485 0.92 ESR2 (0.41) ESR1ESR2LCK
SCHEMBL11050289 0.91 ESR1 (0.39) ESR1ESR2WEE1LCK
SCHEMBL11060337 0.87 CRHR1 (0.33)
SCHEMBL11055393 0.86 ESR1 (0.38) ESR1ESR2
SCHEMBL11055572 0.86 ESR1 (0.38) ESR1ESR2
SCHEMBL11052642 0.86 ESR1 (0.38) ESR1ESR2WEE1
SCHEMBL11058230 0.85 ESR1 (0.35) ESR1ESR2WEE1LCK
SCHEMBL11053272 0.85 NOS3 (0.32)
SCHEMBL11474313 0.82 MEN1 (0.31)
SCHEMBL11050393 0.81 ESR1 (0.31) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed