SCHEMBL11056404

SCHEMBL11056404

CCc1cccc(CC)c1NC(=N)NC(=O)Nc1c(C)cccc1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 2/20 0.54
SCN5A Q14524 2/20 0.54
POLB P06746 3/20 0.51
DRD2 P14416 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2B P41595 1/20 0.50
PKM P14618 1/20 0.49
NLRP3 Q96P20 1/20 0.47
ALDH1A1 P00352 3/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ALOX12 P18054 1/20 0.46
ATM Q13315 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PTGS2 P35354 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11274843 0.91 ALDH1A1 (0.50) CACNA1CSCN5APOLBNLRP3ALDH1A1
SCHEMBL11278731 0.89 POLB (0.62) SCN5APOLBDRD2HTR2AHTR2B
SCHEMBL10615584 0.87 CACNA1C (0.52) CACNA1CSCN5APOLBDRD2HTR2A
SCHEMBL11252413 0.83 POLB (0.51) POLBNLRP3ALDH1A1HTTSMN1; SMN2
SCHEMBL10939937 0.83 CACNA1C (0.61) CACNA1CSCN5ANLRP3ALDH1A1HTT
SCHEMBL9177252 0.82 ALDH1A1 (0.57) POLBNLRP3ALDH1A1HTTSMN1; SMN2
SCHEMBL6698675 0.82 NLRP3 (0.50) CACNA1CSCN5APOLBDRD2HTR2A
SCHEMBL7169954 0.82 CACNA1C (0.57) CACNA1CSCN5APOLBDRD2HTR2A
Hydrochloric Acid SCHEMBL11437019 0.82 CACNA1C (0.60) CACNA1CSCN5APKMNLRP3ALDH1A1
SCHEMBL11058401 0.82 POLB (0.54) POLBDRD2HTR2AHTR2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed