SCHEMBL11056545

SCHEMBL11056545

CCc1cc(CC)c(NC(=O)NC(=N)NC)c(CC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 4/20 0.42
CACNA1C Q13936 3/20 0.42
PLK1 P53350 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HSPA5 P11021 1/20 0.32
MTNR1A P48039 1/20 0.31
ANPEP P15144 1/20 0.31
AKT1 P31749 1/20 0.31
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
RAB9A P51151 1/20 0.30
F2 P00734 1/20 0.30
PLG P00747 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11057721 0.88 ALDH1A1 (0.41) SCN5ACACNA1CPLK1MEN1KMT2A
SCHEMBL11286922 0.87 SCN5A (0.34) SCN5ACACNA1CPLK1MEN1GAA
Hydrochloric Acid SCHEMBL11505153 0.85 SCN5A (0.43) SCN5ACACNA1CALDH1A1KDM4ELMNA
SCHEMBL10903898 0.84 SCN5A (0.41) SCN5ACACNA1CMEN1KMT2AKDM4E
SCHEMBL11060263 0.83 ALDH1A1 (0.36) MEN1GAAKMT2AALDH1A1KDM4E
SCHEMBL10939937 0.83 CACNA1C (0.61) SCN5ACACNA1CALDH1A1KDM4ELMNA
SCHEMBL11407438 0.83 SCN5A (0.47) SCN5ACACNA1CMEN1GAAKMT2A
SCHEMBL10946655 0.82 SCN5A (0.41) SCN5ACACNA1CPLK1MEN1KMT2A
SCHEMBL10906414 0.82 SCN5A (0.41) SCN5ACACNA1CMEN1GAAKMT2A
SCHEMBL10906933 0.82 SCN5A (0.39) SCN5ACACNA1CKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed