SCHEMBL11057271

SCHEMBL11057271

COc1ccc(-c2nc(S)n(CCO)c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
PTGS2 P35354 2/20 0.41
LMNA P02545 5/20 0.41
NPSR1 Q6W5P4 4/20 0.41
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 3/20 0.41
HTT P42858 3/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 1/20 0.39
HIF1A Q16665 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5443200 0.79 ALDH1A1 (0.47) MEN1KMT2APTGS2LMNANPSR1
SCHEMBL8008240 0.71 KDM4E (0.63) LMNANPSR1ALDH1A1KDM4EL3MBTL1
SCHEMBL7995686 0.71 TEK (0.58) MEN1KMT2ALMNANPSR1ALDH1A1
SCHEMBL10964771 0.70 MEN1 (0.48) MEN1KMT2APTGS2ALDH1A1MAPT
SCHEMBL7996428 0.69 KDM4E (0.53) LMNANPSR1ALDH1A1KDM4EL3MBTL1
SCHEMBL6177031 0.69 MAPK14 (0.69)
SCHEMBL11057267 0.68 ALDH1A1 (0.42) MEN1KMT2APTGS2LMNANPSR1
SCHEMBL10989518 0.67 ALDH1A1 (0.47) MEN1KMT2ALMNANPSR1ALDH1A1
SCHEMBL11169683 0.67 KMT2A (0.44) MEN1KMT2APTGS2LMNANPSR1
SCHEMBL11016914 0.66 KMT2A (0.43) MEN1KMT2APTGS2LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440776-A ANTIARTHRITIC AGENTS; ANTIALLERGENS; BRONCHODILATOR AGENTS; SKIN DORDERS SCHERING AKTIENGESELLSCHAFT (DE) 1984-04-03 US disclosed
US-4355039-A Antiinflammatory-4,5-diaryl-2-substituted-thio-imidazoles and their corresponding sulfoxides and sulfones SCHERING, AKTIENGESELLSCHAFT (DE) 1982-10-19 US disclosed
US-4269847-A ANTIALLERGENS; DERIVATIVES OF 4,5-BIS/PHENYL-2-MERCAPTO-, THIO-, S SCHERING AKTIENGESELLSCHAFT (DE) 1981-05-26 US disclosed