SCHEMBL11060104

SCHEMBL11060104

CNC(=N)NC(=S)Nc1c(C)cc(C)cc1C

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 7/20 0.49
LMNA P02545 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGD P15428 2/20 0.39
RAPGEF4 Q8WZA2 1/20 0.38
QPCT Q16769 2/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
AKT1 P31749 2/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11137127 0.86 ALDH1A1 (0.49) KDM4EALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL11277645 0.84 ALDH1A1 (0.53) KDM4EALDH1A1LMNAHPGDRAPGEF4
SCHEMBL11058243 0.83 LMNA (0.49) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
SCHEMBL11511410 0.81 ALDH1A1 (0.59) KDM4EALDH1A1LMNASMN1; SMN2RAPGEF4
SCHEMBL11055416 0.81 KDM4E (0.50) KDM4EALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL11051094 0.79 ALDH1A1 (0.58) ALDH1A1LMNAHPGDMEN1KMT2A
SCHEMBL15484217 0.79 KDM4E (0.63) KDM4EALDH1A1LMNASMN1; SMN2RAPGEF4
SCHEMBL11134286 0.75 ALDH1A1 (0.37) KDM4EALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL11133351 0.73 ALDH1A1 (0.35) KDM4EALDH1A1LMNASMN1; SMN2HPGD
Hydrochloric Acid SCHEMBL11141191 0.72 GAA (0.60) ALDH1A1LMNASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed